209. Nickel-Catalyzed Negishi Arylations of Propargylic Bromides: A  Mechanistic Investigation
Schley, N. D.; Fu, G. C. 
J. Am. Chem. Soc.  2014, 136, 16588–16593.
208. Biphenyl-Derived Phosphepines as Chiral Nucleophilic Catalysts: Enantioselective [4+1] Annulations To Form Functionalized Cyclopentenes
Ziegler, D. T.; Riesgo, L.; Ikeda, T.; Fujiwara, Y.; Fu, G. C. 
Angew. Chem. Int. Ed. 2014, 53, 13183–13187.
207. Stereoconvergent Arylations and Alkenylations of Unactivated Alkyl Electrophiles: Catalytic Enantioselective Synthesis of Secondary Sulfonamides and Sulfones
Choi, J.; Martín-Gago, P.; Fu, G. C. 
J. Am. Chem. Soc. 2014, 136, 12161–12165.
206. Enantioselective Nucleophile-Catalyzed Synthesis of Tertiary Alkyl Fluorides via the α-Fluorination of Ketenes: Synthetic and Mechanistic Studies
Lee, S. Y.; Neufeind, S.; Fu, G. C. 
J. Am. Chem. Soc. 2014, 136, 8899–8902.
205. Oxygen Nucleophiles as Reaction Partners in Photoinduced, Copper-Catalyzed Cross-Couplings: O-Arylations of Phenols at Room Temperature
Tan, Y.; Muñoz-Molina, J. M.; Fu, G. C.; Peters, J. C.  
Chem. Sci. 2014, 5, 2831–3835.
204. Catalytic Asymmetric Synthesis of Tertiary Alkyl Fluorides: Negishi Cross-Couplings of Racemic α,α-Dihaloketones
Liang, Y.; Fu, G. C.
J. Am. Chem. Soc. 2014, 136, 5520–5524.
203. Catalytic Enantioselective Cyclization/Cross-Coupling with Alkyl Electrophiles
Cong, H.; Fu, G. C.
J. Am. Chem. Soc. 2014, 136, 3788–3791.
202. Photoinduced, Copper-Catalyzed Alkylation of Amides with Unactivated Secondary Alkyl Halides at Room Temperature
Do, H.-Q.; Bachman, S.; Bissember, A. C.; Peters, J. C.; Fu, G. C.
J. Am. Chem. Soc. 2014, 136, 2162–2167.
201. Nickel/Bis(oxazoline)-Catalyzed Asymmetric Negishi Arylations of Racemic Secondary Benzylic Electrophiles to Generate Enantioenriched 1,1-Diarylalkanes
Do, H.-Q.; Chandrashekar, E. R. R.; Fu, G. C.
J. Am. Chem. Soc. 2013, 135, 16288–16291.
200. A Versatile Approach to Ullmann C–N Couplings at Room Temperature: New Families of Nucleophiles and Electrophiles for Photoinduced, Copper-Catalyzed Processes
Ziegler, D. T.; Choi, J.; Muñoz-Molina, J. M.; Bissember, A. C.; Peters, J. C.; Fu, G. C.
J. Am. Chem. Soc. 2013, 135, 13107–13112.
199. Enantioconvergent Cross-Couplings of Racemic Alkylmetal Reagents with Unactivated Secondary Alkyl Electrophiles: Catalytic Asymmetric Negishi α-Alkylations of N-Boc-pyrrolidine
Cordier, C. J.; Lundgren, R. J.; Fu, G. C.
J. Am. Chem. Soc. 2013, 135, 10946–10949.
198. A New Family of Nucleophiles for Photoinduced, Copper-Catalyzed Cross-Couplings via Single-Electron Transfer: Reactions of Thiols with Aryl Halides Under Mild Conditions (0 °C)
Uyeda, C.; Tan, Y.; Fu, G. C.; Peters, J. C.
J. Am. Chem. Soc. 2013, 135, 9548–9552.
197. Transition-Metal-Catalyzed Alkylations of Amines with Alkyl Halides: Photoinduced, Copper-Catalyzed Couplings of Carbazoles
Bissember, A. C.; Lundgren, R. J.; Creutz, S. E.; Peters, J. C.; Fu, G. C.
Angew. Chem. Int. Ed. 2013, 52, 5129–5133.
196. Nickel-Catalyzed Carbon–Carbon Bond-Forming Reactions of Unactivated Tertiary Alkyl Halides: Suzuki Arylations
Zultanski, S.; Fu, G. C.
J. Am. Chem. Soc. 2013, 135, 624–627.
195. Catalytic Asymmetric C–N Bond Formation: Phosphine-Catalyzed Intra- and Intermolecular γ-Addition of Nitrogen Nucleophiles to Allenoates and Alkynoates
Lundgren, R. J.; Wilsily, A.; Marion, N.; Ma, C.; Chung, Y. K.; Fu, G. C. 
Angew. Chem. Int. Ed. 2013, 52, 2525–2528.
194. Photoinduced Ullmann C–N Coupling: Demonstrating the Viability of a Radical Pathway 
Creutz, S. E.; Lotito, K. J.; Fu, G. C.; Peters, J. C. 
​Science 2012, 338, 647–651.
193. Catalytic Enantioselective Cross-Couplings of Secondary Alkyl Electrophiles with Secondary Alkylmetal Nucleophiles: Negishi Reactions of Racemic Benzylic Bromides with Achiral Alkylzinc Reagents
Binder, J. T.; Cordier, C. J.; Fu, G. C.
J. Am. Chem. Soc. 2012, 134, 17003–17006.
192. Nonenzymatic Dynamic Kinetic Resolution of Secondary Alcohols via Enantioselective Acylation: Synthetic and Mechanistic Studies
Lee, S. Y.; Murphy-Knight, J. M.; Ukai, A.; Fu, G. C.
J. Am. Chem. Soc. 2012, 134, 15149–15153.
191. A Mild, Palladium-Catalyzed Method for the Dehydrohalogenation of Alkyl Bromides: Synthetic and Mechanistic Studies
Bissember, A. C.; Levina, A.; Fu, G. C.
J. Am. Chem. Soc. 2012, 134, 14232–14237.
190. Nickel-Catalyzed Coupling Reactions of Alkyl Electrophiles, Including Unactivated Tertiary Halides, To Generate Carbon–Boron Bonds
Dudnik, A. S.; Fu, G. C.
J. Am. Chem. Soc. 2012, 134, 10693–10697.
189. Catalytic Asymmetric Synthesis of Secondary Nitriles via Stereoconvergent Negishi Arylations and Alkenylations of Racemic α-Bromonitriles
Choi, J.; Fu, G. C.
J. Am. Chem. Soc. 2012, 134, 9102–9105.
188. New Directing Groups for Metal-Catalyzed Asymmetric Carbon–Carbon Bond-Forming Processes: Stereoconvergent Alkyl–Alkyl Suzuki Cross-Couplings of Unactivated Electrophiles
Wilsily, A.; Tramutola, F.; Owston, N. A.; Fu, G. C.
J. Am. Chem. Soc. 2012, 134, 5794–5797.
187. Competitive Activity-Based Protein Profiling Identifies Aza-β-Lactams as a Versatile Chemotype for Serine Hydrolase Inhibition
Zuhl, A. M.; Mohr, J. T.; Bachovchin, D. A.; Niessen, S.; Hsu, K.-L.; Berlin, J. M.; Dochnahl, M.; López-Alberca, M. P.; Fu, G. C.; Cravatt, B. F.
J. Am. Chem. Soc. 2012, 134, 5068–5071.
186. Nickel-Catalyzed Enantioselective Cross-Couplings of Racemic Secondary Electrophiles That Bear an Oxygen Leaving Group
Oelke, A. J.; Sun, J.; Fu, G. C.
J. Am. Chem. Soc. 2012, 134, 2966–2999.
185. Catalytic Asymmetric γ-Alkylation of Carbonyl Compounds via Stereoconvergent Suzuki Cross-Couplings
Zultanski, S. L.; Fu, G. C.
J. Am. Chem. Soc. 2011, 133, 15362–15364.
184. Enantioselective carbon–sulfur bond formation: γ additions of arylthiols to allenoates catalyzed by a chiral phosphepine
Fujiwara, Y.; Sun, J.; Fu, G. C.
Chem. Sci. 2011, 2, 2196–2198.
183. Application of a New Chiral Phosphepine to the Catalytic Asymmetric Synthesis of Highly Functionalized Cyclopentenes That Bear an Array of Heteroatom-Substituted Quaternary Stereocenters
Fujiwara, Y.; Fu, G. C.
J. Am. Chem. Soc. 2011, 133, 12293–12297.
182. Stereoconvergent Amine-Directed Alkyl–Alkyl Suzuki Reactions of Unactivated Secondary Alkyl Chlorides
Lu, Z.; Wilsily, A.; Fu, G. C.
J. Am. Chem. Soc. 2011, 133, 8154–8157.
181. Academic cross-fertilization by public screening yields a remarkable class of protein phosphatase methylesterase-1 inhibitors
Bachovchin, D. A.; Mohr, J. T.; Speers, A. E.; Wang, C.; Berlin, J. M.; Spicer, T. P.; Fernandez-Vega, V.; Chase, P.; Hodder, P. S.; Schurer, S.; Nomura, D. K.; Rosen, H.; Fu, G. C.; Cravatt, B. F.
Proc. Natl. Acad. Sci. U.S.A. 2011, 108, 6811–6816.
180. Phosphine-catalyzed asymmetric additions of malonate esters to γ-substituted allenoates and allenamides
Sinisi, R.; Sun, J.; Fu, G. C.
Proc. Natl. Acad. Sci. U.S.A. 2010, 107, 20652–20654. 
179. Asymmetric Alkyl−Alkyl Cross-Couplings of Unactivated Secondary Alkyl Electrophiles: Stereoconvergent Suzuki Reactions of Racemic Acylated Halohydrins
Owston, N. A.; Fu, G. C.
J. Am. Chem. Soc. 2010, 132, 11908–11909.
178. Asymmetric Suzuki Cross-Couplings of Activated Secondary Alkyl Electrophiles: Arylations of Racemic α-Chloroamides
Lundin, P.; Fu, G. C.
J. Am. Chem. Soc. 2010, 132, 11027–11029.
177. Alkyl–Alkyl Suzuki Cross-Coupling of Unactivated Secondary Alkyl Chlorides
Lu, Z.; Fu, G. C.
Angew. Chem., Int. Ed. 2010, 49, 6676–6678.
176. Nickel-Catalyzed Enantioselective Negishi Cross-Couplings of Racemic Secondary α-Bromo Amides with Alkylzinc Reagents
Lou, S.; Fu, G. C.
Org. Synth. 2010, 87, 330–338.
175. Nickel-Catalyzed Asymmetric Negishi Cross-Couplings of Racemic Secondary Allylic Chlorides with Alkylzincs 
Lou, S.; Fu, G. C.
Org. Synth. 2010, 87, 317–329.
174. Synthesis of Chiral Pyridine Bis(Oxazoline) Ligands for Nickel-Catalyzed Asymmetric Negishi Cross-Couplings of Secondary Allylic Chlorides with Alkylzincs
Lou, S.; Fu, G. C.
Org. Synth. 2010, 87, 310–316.
173. Palladium-Catalyzed Alkyl–Alkyl Suzuki Cross-Couplings of Primary Alkyl Bromides at Room Temperature 
Lou, S.; Fu, G. C.
Org. Synth. 2010, 87, 299–309.
172. Pd/P(t-Bu)3-Catalyzed Suzuki Cross-Couplings in the Presence of Water 
Lou, S.; Fu, G. C.
Adv. Synth. Catal. 2010, 352, 2081–2084.
171. Enantioselective Alkenylation via Nickel-Catalyzed Cross-Coupling with Organozirconium Reagents 
Lou, S.; Fu, G. C.
J. Am. Chem. Soc. 2010, 132, 5010–5011.
170. Phosphine-Catalyzed Formation of Carbon–Sulfur Bonds: Catalytic Asymmetric Synthesis of γ-Thioesters 
Sun, J.; Fu, G. C.
J. Am. Chem. Soc. 2010, 132, 4568–4569.
169. Applications of Aza- and Phosphaferrocenes and Related Compounds in Asymmetric Catalysis 
Chiral Ferrocenes in Asymmetric Catalysis; Dai, L.-X., Hou, X.-L., Ed.; Wiley–VCH: New York, 2010; Chapter 11.
Marion, N. M.; Fu. G. C.

168. Nickel/Bis(oxazoline)-Catalyzed Asymmetric Kumada Reactions of Alkyl Electrophiles: Cross- Couplings of Racemic α-Bromoketones
Lou, S.; Fu, G. C.
J. Am. Chem. Soc. 2010, 132, 1264–1266.
167. Phosphine-Catalyzed Stereoselective Synthesis of Highly Functionalized Diquinanes 
Wilson, J. E.; Sun, J.; Fu, G. C.
Angew. Chem., Int. Ed. 2010, 49, 161–163.

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